Zamicastat

• Catalog Number: orb1308925
• Category: Small Molecules
• Description: Zamicastat
• CAS Number: 1080028-80-3
• Purity: 98.43%
• MW: 401.47
• SMILES: C(CNCC1=CC=CC=C1)C=2N([C@@H]3CC=4C(OC3)=C(F)C=C(F)C4)C(=S)NC2
• Formula: C₂₁H₂₁F₂N₃OS
• Biological Activity: Zamicastat (BIA 5-1058) is an inhibitor of dopamine β-hydroxylase (DBH), and is also a concentration-dependent dual inhibitor of P-gp and BCRP(IC50 values of 73.8 μM and 17.0 μM, respectively).
• Storage: Store at -20°C for 12 months.
• Note: For research use only
• Expiration Date: 12 months from date of receipt.