YKL-5-124

• Catalog Number: orb1305905
• Category: Small Molecules
• Description: YKL-5-124
• CAS Number: 1957203-01-8
• Purity: 99.50%
• MW: 515.61
• SMILES: N(C(=O)C1=CC=C(NC(C=C)=O)C=C1)C=2C3=C(C(C)(C)N(C(N[C@H](CN(C)C)C4=CC=CC=C4)=O)C3)NN2
• Formula: C₂₈H₃₃N₇O₃
• Biological Activity: YKL-5-124, a potent, selective and covalent CDK7 inhibitor with an IC50 of 9.7 nM, 1300 nM and 3020 nM for CDK7/Mat1/CycH, CDK2 and CDK9 respectively, displays biochemical and cellular selectivity for CDK7 over CDK12/13.
• Storage: Store at -20°C for 12 months.
• Note: For research use only
• Expiration Date: 12 months from date of receipt.