YAP-TEAD Inhibitor 1 (Peptide 17)

• Catalog Number: orb654735
• Category: Small Molecules
• Description: YAP-TEAD Inhibitor 1 (Peptide 17)
• CAS Number: 1659305-79-9
• Purity: > 98%
• MW: 2133.88
• SMILES: C(F)(F)(F)C(=O)O.C(N1CCC[C@H]1C(=O)N[C@H](C(=O)N)CCC(=O)O)([C@@H]1CCCN1C(=O)[C@H](CCCCN)NC(C1CSSCC[C@@H](C(N[C@H](C(N[C@H](C(N[C@H](C(=O)N[C@@]([H])(CCCC)C(=O)N2CCC[C@@]2([H])C(=O)N[C@@H](C)C(=O)N[C@@]([H])(CO)C(=O)N[C@@H](CC2C=CC=CC=2)C(=O)N1)CCCCN)=O)CCCNC(N)=N)=O)CC(C)C)=O)NC(=O)[C@H](CC1C=CC=C(Cl)C=1)NC([C@@H]1CCCN1C(=O)[C@H](C(C)C)NC(=O)C)=O)=O)=O
• Formula: C₉₅H₁₄₅ClF₃N₂₃O₂₃S₂
• Storage: 2 years -20°C Powder, 2 weeks4°C in DMSO,6 months-80°C in DMSO
• Alternative names: YAP-TEAD-IN-1 TFA;YAP-TEAD (Peptide 17).TFA;(S)-4-
• Background: YAP-TEAD-IN-1 TFA is a potent and competitive peptide inhibitor of?YAP-TEAD interaction (IC50=25 nM). YAP-TEAD-IN-1 TFA is a 17mer peptide and shows a higher the binding affinity to TEAD1 (Kd=15 nM) than YAP (50-171) (Kd= 40 nM)
• Note: For research use only
• Expiration Date: 12 months from date of receipt.

CAS no: 1659305-79-9