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Catalog Number | orb1296112 |
---|---|
Category | Small Molecules |
Description | UNC0646 |
CAS Number | 1320288-17-2 |
Purity | 100% |
MW | 621.9 |
SMILES | N(C=1C2=C(N=C(N1)N3CCN(C(C)C)CCC3)C=C(OCCCN4CCCCC4)C(OC)=C2)C5CCN(CC5)C6CCCCC6 |
Formula | C36H59N7O2 |
Biological Activity | UNC0646 is a potent and selective inhibitor of the homologous protein lysine methyltransferases, G9a and GLP (IC50s: 6 nM/15 nM for G9a/GLP). UNC0646(UNC 0646) potently blocks G9a/GLP methyltransferase activity in cells (IC50: 10 nM in MCF7 cells); exhibits low cellular toxicity (EC50: 4.7 μM in MCF7 cells). |
Storage | Store at -20°C for 12 months. |
Note | For research use only |
Expiration Date | 12 months from date of receipt. |
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