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TGR5 Receptor Agonist 4

TGR5 Receptor Agonist 4

Catalog Number: orb1943763

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Catalog Numberorb1943763
CategorySmall Molecules
DescriptionTGR5 Receptor Agonist 4, a selective agonist for the Bile Acid Receptor (TGR5), exhibits potent activity with an EC50 of 2 nM for human TGR5 (hTGR5) and 3 nM for mouse TGR5 (mTGR5). It is notably involved in mediating hypoglycemic and weight loss effects [1].
CAS Number1872436-42-4
Purity98.00%
MW470.95
SMILESC(OCC1=C(OC)C=CC=C1)(=O)C=2[C@@H](CC(=O)N(C[C@H]3CCCO3)C2C)C=4C=CC(Cl)=NC4
FormulaC25H27ClN2O5
Biological ActivityTGR5 Receptor Agonist 4, a selective agonist for the Bile Acid Receptor (TGR5), exhibits potent activity with an EC50 of 2 nM for human TGR5 (hTGR5) and 3 nM for mouse TGR5 (mTGR5). It is notably involved in mediating hypoglycemic and weight loss effects [1].
Storage-20°C
NoteFor research use only
Expiration Date12 months from date of receipt.
  • TGR5 agonist 4 [orb2277954]

    98.00%

    444.55

    C24H38F2O5

    50 mg, 5 mg
  • TGR5 Receptor Agonist 3 [orb1686487]

    98%

    2643391-08-4

    513.54

    C29H27N3O6

    25 mg, 100 mg, 50 mg