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Catalog Number | orb1943763 |
---|---|
Category | Small Molecules |
Description | TGR5 Receptor Agonist 4 |
CAS Number | 1872436-42-4 |
MW | 470.95 |
SMILES | C(OCC1=C(OC)C=CC=C1)(=O)C=2[C@@H](CC(=O)N(C[C@H]3CCCO3)C2C)C=4C=CC(Cl)=NC4 |
Formula | C25H27ClN2O5 |
Biological Activity | TGR5 Receptor Agonist 4, a selective agonist for the Bile Acid Receptor (TGR5), exhibits potent activity with an EC50 of 2 nM for human TGR5 (hTGR5) and 3 nM for mouse TGR5 (mTGR5). It is notably involved in mediating hypoglycemic and weight loss effects [1]. |
Note | For research use only |
Expiration Date | 12 months from date of receipt. |
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