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    TGR5 Receptor Agonist 4

    TGR5 Receptor Agonist 4

    Catalog Number: orb1943763

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    Catalog Numberorb1943763
    CategorySmall Molecules
    DescriptionTGR5 Receptor Agonist 4
    CAS Number1872436-42-4
    MW470.95
    SMILESC(OCC1=C(OC)C=CC=C1)(=O)C=2[C@@H](CC(=O)N(C[C@H]3CCCO3)C2C)C=4C=CC(Cl)=NC4
    FormulaC25H27ClN2O5
    Biological ActivityTGR5 Receptor Agonist 4, a selective agonist for the Bile Acid Receptor (TGR5), exhibits potent activity with an EC50 of 2 nM for human TGR5 (hTGR5) and 3 nM for mouse TGR5 (mTGR5). It is notably involved in mediating hypoglycemic and weight loss effects [1].
    NoteFor research use only
    Expiration Date12 months from date of receipt.
    • TGR5 Receptor Agonist 3 [orb1686487]

      98%

      2643391-08-4

      513.54

      C29H27N3O6

      25 mg, 100 mg, 50 mg
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