Relugolix (TAK-385)

• Catalog Number: orb573025
• Category: Small Molecules
• Description: Relugolix is a novel, non-peptide, orally active gonadotropin-releasing hormone (GnRH) antagonist with IC50 of 0.33 nM in the presence of 40% fetal bovine serum, TAK-385 possesses higher affinity and potent antagonistic activity compared with TAK-013.
• CAS Number: [737789-87-6]
• MW: 623.63
• SMILES: O=C(NOC)NC1=CC=C(C(S2)=C(CN(C)C)C(C(N3C4=NN=C(OC)C=C4)=O)=C2N(CC5=C(F)C=CC=C5F)C3=O)C=C1
• Formula: C₂₉H₂₇F₂N₇O₅S
• Note: For research use only
• Expiration Date: 12 months from date of receipt.