PROTAC BET degrader-2

• Catalog Number: orb572923
• Category: Small Molecules
• Description: PROTAC BET degrader-2 is a highly potent degrader of Bromodomain and Extra-Terminal (BET) proteins with an IC50 value of 9.6 nM in cell growth inhibition in the RS4;11 cells and capable of achieving tumor regression.
• CAS Number: [2093388-33-9]
• MW: 770.84
• SMILES: O=C(C1=NC(NC2=CC(C3CC3)=NN2CC)=C4C(NC5=C4C=C(OC)C(C6=C(C)ON=C6C)=C5)=N1)NCCCC7=CC=CC8=C7CN(C(CC9)C(NC9=O)=O)C8=O
• Formula: C₄₁H₄₂N₁₀O₆
• Note: For research use only
• Expiration Date: 12 months from date of receipt.