Pasireotide (diaspartate)

• Catalog Number: orb1982174
• Category: Small Molecules
• Description: Pasireotide diaspartate (SOM230), a long-acting cyclohexapeptide and somatostatin analog, enhances agonist activity across somatostatin receptor subtypes (sst1/2/3/4/5, with pK i values of 8.2, 9.0, 9.1, < 7.0, and 9.9, respectively). This compound demonstrates antisecretory, antiproliferative, and proapoptotic activities [1] [2].
• CAS Number: 1421446-02-7
• Purity: 98.00%
• MW: 1313.41
• SMILES: OC(C[C@H](N)C(O)=O)=O.O=C1N2[C@@](C(N[C@@H](C3=CC=CC=C3)C(N[C@@H](C(N[C@H](C(N[C@H](C(N[C@H]1CC4=CC=CC=C4)=O)CC5=CC=C(C=C5)OCC6=CC=CC=C6)=O)CCCCN)=O)CC7=CNC8=CC=CC=C78)=O)=O)([H])C[C@H](C2)OC(NCCN)=O.OC(C[C@H](N)C(O)=O)=O
• Formula: C₆₆H₈₀N₁₂O₁₇
• Biological Activity: Pasireotide diaspartate (SOM230), a long-acting cyclohexapeptide and somatostatin analog, enhances agonist activity across somatostatin receptor subtypes (sst1/2/3/4/5, with pK i values of 8.2, 9.0, 9.1, < 7.0, and 9.9, respectively). This compound demonstrates antisecretory, antiproliferative, and proapoptotic activities [1] [2].
• Storage: -20°C
• Note: For research use only
• Expiration Date: 12 months from date of receipt.