OTS186935 trihydrochloride

• Catalog Number: orb746452
• Category: Small Molecules
• Description: OTS186935 trihydrochloride is a protein methyltransferase SUV39H2 inhibitor with an IC50 of 6.49 nM. OTS186935 trihydrochloride shows significant inhibition of tumor growth in mouse xenograft models without any detectable toxicity. OTS186935 trihydrochloride regulates the production of γ-H2AX in cancer cells[1].
• CAS Number: [2093401-85-3]
• MW: 573.34
• SMILES: N1(C2C=CN3C=C(C4=CC(Cl)=C(OC)C=C4OC)N=C3C=2)CC[C@@H](NCC2C=CN=CC=2)C1.Cl.Cl.Cl
• Formula: C₂₅H₂₉Cl₄N₅O₂
• Note: For research use only
• Expiration Date: 12 months from date of receipt.