Omipalisib (GSK-458)

• Catalog Number: orb181012
• Category: Small Molecules
• Description: GSK2126458 is a highly selective and potent inhibitor of PI3K with Ki of 0.019 nM/0.13 nM/0.024 nM/0.06 nM and 0.18 nM/0.3 nM for p110α/β/δ/γ, mTORC1/2 , respectively.
• CAS Number: [1086062-66-9]
• MW: 505.496
• SMILES: S(C1C([H])=C([H])C(=C([H])C=1F)F)(N([H])C1=C(N=C([H])C(=C1[H])C1C([H])=C([H])C2C(=C(C([H])=C([H])N=2)C2=C([H])N=NC([H])=C2[H])C=1[H])OC([H])([H])[H])(=O)=O
• Formula: C₂₅H₁₇F₂N₅O₃S
• Note: For research use only
• Expiration Date: 12 months from date of receipt.