MRK-016

• Catalog Number: orb611735
• Category: Small Molecules
• Description: A potent, functionally selective, CNS-penetrating and orally bioavailable inverse agonist of benzodiazepine site of GABAA α5 receptor with Ki of 0.8-1.5 nM for α1-, α2-, α3-, andα5-containing GABAA receptors.
• CAS Number: [342652-67-9]
• MW: 368.3931
• SMILES: CN1C(COC2C(C(C)(C)C)=C3N(C(=NN=C3)C3C=C(C)ON=3)N=2)=NC=N1
• Formula: C₁₇H₂₀N₈O₂
• Note: For research use only
• Expiration Date: 12 months from date of receipt.