MCH(human, mouse, rat) TFA

• Catalog Number: orb1981608
• Category: Small Molecules
• Description: MCH (human, mouse, rat) TFA is a potent peptide agonist for MCH receptors, exhibiting binding IC50 values of 0.3 nM for MCH1R and 1.5 nM for MCH2R. It is particularly effective against MCH-2R in a CHO cell line, with functional activation EC50 values of 3.9 nM for MCH-1R and 0.1 nM for MCH-2R, as evidenced by intracellular calcium mobilization measured with FLIPR [1].
• Purity: 98.00%
• MW: 2500.86
• Formula: C₁₀₇H₁₆₁F₃N₃₀O₂₈S₄
• Biological Activity: MCH (human, mouse, rat) TFA is a potent peptide agonist for MCH receptors, demonstrating strong affinity with binding IC 50 values of 0.3 nM for MCH1R and 1.5 nM for MCH2R. It is notably effective against MCH-2R in a CHO cell line, as evidenced by the mobilization of intracellular calcium measured with FLIPR, revealing functional activation EC 50 values of 3.9 nM for MCH-1R and 0.1 nM for MCH-2R [1].
• Storage: -20°C
• Note: For research use only
• Expiration Date: 12 months from date of receipt.