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Catalog Number | orb1982696 |
---|---|
Category | Small Molecules |
Description | LAS190792 |
CAS Number | 1347232-69-2 |
MW | 811.36 |
SMILES | COc1cc(NC(=O)OCCN(C)[C@H]2CC[C@@H](CC2)OC(=O)C(O)(c2cccs2)c2cccs2)c(Cl)cc1CNC[C@H](O)c1ccc(O)c2[nH]c(=O)ccc12 |
Formula | C39H43ClN4O9S2 |
Biological Activity | LAS190792 (AZD8999) is a dual-action chemical compound that simultaneously acts as a strong muscarinic antagonist and β2-adrenoceptor agonist. It exhibits significant potency across a range of receptors, with pIC50 values of 8.9 for M1, 8.8 for M2, 8.8 for M3, 9.2 for M4, 8.2 for M5, 7.5 for β1, 9.1 for β2, and 5.6 for β3. Its effectiveness across these receptors makes LAS190792 a viable candidate for bronchodilator applications [1]. |
Note | For research use only |
Expiration Date | 12 months from date of receipt. |
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