KDM5A-IN-1

• Catalog Number: orb1707141
• Category: Small Molecules
• Description: KDM5A-IN-1
• CAS Number: 1905481-36-8
• Purity: 98%
• MW: 290.36
• SMILES: C(=O)(C=1C=C(C(C)C)NN1)N2C[C@H](NC(=O)C3CC3)CC2
• Formula: C₁₅H₂₂N₄O₂
• Biological Activity: KDM5A-IN-1 is an orally available, potent and selective inhibitor of the pan-histidine lysine demethylase 5 KDM5, inhibiting KDM5A, KDM5B, and KDM5C with IC50 values of 45 nM, 56 nM, and 55 nM, respectively.KDM5A-IN-1 inhibits PC9 H3K4Me3, and may be useful in cancer research.
• Note: For research use only
• Expiration Date: 12 months from date of receipt.