HJC0197

• Catalog Number: orb692047
• Category: Small Molecules
• Description: HJC0197 is a potent Epac1 (exchange protein directly activated by cAMP 1) and Epac2 (IC50=5.9 μM for Epac2) antagonist. HJC0197 selectively blocks cAMP-induced Epac activation. HJC0197 inhibits Epac1-mediated Rap1-GDP exchange activity at 25 μM in the presence of equal concentration of cAMP.
• CAS Number: [1383539-73-8]
• MW: 339.45
• SMILES: N#CC1C(=O)NC(SCC2C(C)=CC=C(C)C=2)=NC=1C1CCCC1
• Formula: C₁₉H₂₁N₃OS
• Note: For research use only
• Expiration Date: 12 months from date of receipt.