GSK2798745

• Catalog Number: orb1707241
• Category: Small Molecules
• Description: GSK2798745
• CAS Number: 1419609-94-1
• MW: 460.53
• SMILES: C([C@]1(C)C[C@]2(CN(C(=O)O2)C=3C=NC(C(C)(C)O)=CN3)CCC1)N4C=5C(N=C4)=CC=C(C#N)C5
• Formula: C₂₅H₂₈N₆O₃
• Biological Activity: GSK2798745 is an orally active transient receptor potential vanilloid 4 (TRPV4) ion channel blocker (IC50s: 1.8 and 1.6 nM for hTRPV4 and rTRPV4). It is used in research for the treatment of pulmonary edema associated with congestive heart failure.
• Note: For research use only
• Expiration Date: 12 months from date of receipt.