GSK-2807 free base

• Catalog Number: orb1739742
• Category: Small Molecules
• Description: GSK-2807 free base
• CAS Number: 2245255-65-4
• Purity: 0.98
• MW: 452.51
• SMILES: O[C@H]1[C@H](N2C=3C(N=C2)=C(N)N=CN3)O[C@H](CN(CC[C@@H](C(O)=O)N)CCCN(C)C)[C@H]1O
• Formula: C₁₉H₃₂N₈O₅
• Biological Activity: GSK2807 is a potent and selective, SAM-competitive inhibitor of SMYD3 (Ki = 14 nM). GSK2807 bridges the gap between the SAM-binding pocket and the substrate lysine tunnel of SMYD3. GSK2807 may be useful for cancer treatment.
• Note: For research use only
• Expiration Date: 12 months from date of receipt.