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Catalog Number | orb1688748 |
---|---|
Category | Small Molecules |
Description | GSK-1070916 |
CAS Number | 942918-07-2 |
Purity | 98.51% |
MW | 507.63 |
SMILES | C(C)N1C=C(C(=N1)C2=CC=C(NC(N(C)C)=O)C=C2)C3=C4C(NC(=C4)C5=CC(CN(C)C)=CC=C5)=NC=C3 |
Formula | C30H33N7O |
Biological Activity | GSK1070916 is a reversible and ATP-competitive inhibitor of Aurora B/C with IC50 of 3.5 nM/6.5 nM. It displays > 100-fold selectivity against the closely related Aurora A-TPX2 complex. Phase 1. |
Note | For research use only |
Expiration Date | 12 months from date of receipt. |
> 98% (HPLC) | |
942918-07-2 |
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