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    GSK-1070916

    GSK-1070916

    Catalog Number: orb1688748

    DispatchUsually dispatched within 3-5 working days
    $ 698.00
    Catalog Numberorb1688748
    CategorySmall Molecules
    DescriptionGSK-1070916
    CAS Number942918-07-2
    Purity98.51%
    MW507.63
    SMILESC(C)N1C=C(C(=N1)C2=CC=C(NC(N(C)C)=O)C=C2)C3=C4C(NC(=C4)C5=CC(CN(C)C)=CC=C5)=NC=C3
    FormulaC30H33N7O
    Biological ActivityGSK1070916 is a reversible and ATP-competitive inhibitor of Aurora B/C with IC50 of 3.5 nM/6.5 nM. It displays > 100-fold selectivity against the closely related Aurora A-TPX2 complex. Phase 1.
    NoteFor research use only
    Expiration Date12 months from date of receipt.
    • GSK-1070916 [orb1223566]

      > 98% (HPLC)

      942918-07-2

      1 g, 500 mg, 200 mg, 5 mg, 10 mg, 25 mg, 50 mg, 100 mg
    • GSK-1070916 [orb181011]

      [942918-07-2]

      507.63

      C30H33N7O

      10 mM * 1 mL in DMSO, 100 mg, 1000 mg, 250 mg
    • GSK-1070916 [orb609887]

      ≥98%

      942918-07-2

      507.63

      C30H33N7O

      1 mg, 10 mg, 5 mg
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