GPR81 agonist 1

• Catalog Number: orb1687388
• Category: Small Molecules
• Description: GPR81 agonist 1
• CAS Number: 1620992-67-7
• Purity: 99.68%
• MW: 446.63
• SMILES: C(C(=O)N1CCN(C)CC1)C2=C(N=C(NC(=O)[C@H]3CC[C@H](C)CC3)S2)C4=CC=CS4
• Formula: C₂₂H₃₀N₄O₂S₂
• Biological Activity: GPR81 agonist 1 is a potent and highly selective GPR81 agonist, with EC 50 s of 58 nM and 50 nM for human and mouse GPR81, respectively. GPR81 agonist 1 inhibits lipolysis in differentiated 3T3-L1 adipocytes. GPR81 agonist 1 suppresses lipolysis in mice without cutaneous flushing. GPR81 agonist 1 displays remarkable selectivity for GPR81 over GPR109a [1].
• Storage: Store at -20°C for 12 months.
• Note: For research use only
• Expiration Date: 12 months from date of receipt.