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Catalog Number | orb1687388 |
---|---|
Category | Small Molecules |
Description | GPR81 agonist 1 |
CAS Number | 1620992-67-7 |
Purity | 99.68% |
MW | 446.63 |
SMILES | C(C(=O)N1CCN(C)CC1)C2=C(N=C(NC(=O)[C@H]3CC[C@H](C)CC3)S2)C4=CC=CS4 |
Formula | C22H30N4O2S2 |
Biological Activity | GPR81 agonist 1 is a potent and highly selective GPR81 agonist, with EC 50 s of 58 nM and 50 nM for human and mouse GPR81, respectively. GPR81 agonist 1 inhibits lipolysis in differentiated 3T3-L1 adipocytes. GPR81 agonist 1 suppresses lipolysis in mice without cutaneous flushing. GPR81 agonist 1 displays remarkable selectivity for GPR81 over GPR109a [1]. |
Storage | Store at -20°C for 12 months. |
Note | For research use only |
Expiration Date | 12 months from date of receipt. |
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