GNE-781

• Catalog Number: orb1308265
• Category: Small Molecules
• Description: GNE-781
• CAS Number: 1936422-33-1
• Purity: 98.73%
• MW: 525.59
• SMILES: C(NC)(=O)N1CC=2C(=NN(C2CC1)C3CCOCC3)N4C=5C(=CC(=C(C(F)F)C5)C6=CN(C)N=C6)CCC4
• Formula: C₂₇H₃₃F₂N₇O₂
• Biological Activity: GNE-781 is a highly potent and selective inhibitor of CBP (IC50: 0.94 nM in TR-FRET assay). GNE-781 also inhibits BRET and BRD4(1) (IC50s: 6.2 nM and 5100 nM, respectively).
• Storage: Store at -20°C for 12 months.
• Note: For research use only
• Expiration Date: 12 months from date of receipt.