GNE-0439

• Catalog Number: orb1709573
• Category: Small Molecules
• Description: GNE-0439
• CAS Number: 1241902-40-8
• Purity: 98%
• MW: 345.48
• SMILES: C(N[C@@H]([C@@H](C)C)C(O)=O)(=O)C1=CC=C(C=C1)C2CCC(CCC)CC2
• Formula: C₂₁H₃₁NO₃
• Biological Activity: GNE-0439 is a novel Nav1.7-selective inhibitor (IC50: 0.34 uM) and inhibits Nav1.5 (IC50: 38.3 μM). GNE-0439 inhibits mutant N1742K channels (IC50: 0.37 uM) in membrane potential assays.
• Note: For research use only
• Expiration Date: 12 months from date of receipt.