GGTI-2418

• Catalog Number: orb1709612
• Category: Small Molecules
• Description: GGTI-2418
• CAS Number: 501010-06-6
• Purity: 99.18%
• MW: 441.52
• SMILES: CC(C)C[C@H](NC(=O)N1CCN(Cc2nc[nH]c2C)C(=O)[C@@H]1Cc1ccccc1)C(O)=O
• Formula: C₂₃H₃₁N₅O₄
• Biological Activity: GGTI-2418 is a highly potent, competitive, and selective inhibitor of geranylgeranyltransferase I (GGTase I), showing inhibitory activities with IC50 values of 9.5 nM for GGTase I and 53 μM for FTase, respectively. Additionally, it enhances p27(Kip1) expression and induces significant regression of breast tumors.
• Storage: -20°C
• Note: For research use only
• Expiration Date: 12 months from date of receipt.