GDC-0810

• Catalog Number: orb611604
• Category: Small Molecules
• Description: GDC-0810 (ARN-810, Brilanestrant) is a non-steroidal, orally bioavailable selective estrogen receptor degrader (SERD) with IC50 of 0.7 nM (ER-α degradation), binds to ERα and ERβ with with Ki of 3.8 and 3.7 nM, respectively.
• CAS Number: [1365888-06-7]
• MW: 446.9006
• SMILES: O=C(C=CC1C=CC(C(=C(CC)C2C(Cl)=CC(F)=CC=2)C2C=CC3NN=CC=3C=2)=CC=1)O
• Formula: C₂₆H₂₀ClFN₂O₂
• Note: For research use only
• Expiration Date: 12 months from date of receipt.