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    FGTI-2734

    FGTI-2734

    Catalog Number: orb757630

    DispatchUsually dispatched within 5-10 working days
    $ 3,856.00
    Catalog Numberorb757630
    CategorySmall Molecules
    DescriptionFGTI-2734 is a RAS C-terminal mimetic dual farnesyl transferase (FT) and geranylgeranyl transferase-1 (GGT-1) inhibitor. It can prevent membrane localization of KRAS, hence solving KRAS resistance problem and thwarting mutant KRAS patient-derived pancreatic tumors.
    CAS Number[1247018-19-4]
    MW510.6324
    SMILESO=S(C1=NC=CC=C1)(N(CC2CCCCC2)CCN(CC3=CN=CN3C)C4=CC=C(C=C4F)C#N)=O
    FormulaC26H31FN6O2S
    NoteFor research use only
    Expiration Date12 months from date of receipt.
    • FGTI-2734 [orb1309674]

      98%

      1247018-19-4

      510.63

      C26H31FN6O2S

      10 mg, 1 mg, 100 mg, 50 mg, 25 mg, 5 mg, 1 mL*10mM (in DMSO)
    • FGTI-2734 [orb1889182]

      1247018-19-4

      50 mg
    • FGTI-2734 [orb1889183]

      1247018-19-4

      5 mg
    • FGTI-2734 [orb1889184]

      1247018-19-4

      10 mg
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