EST73502

• Catalog Number: orb1910393
• Category: Small Molecules
• Description: EST73502 is a selective, orally active and blood-brain barrier (BBB) penetrant dual μ-opioid receptor (MOR) agonist and σ1 receptor (σ1R) antagonist, with Kis of 64 nM and 118 nM for MOR and σ1R, respectively. EST73502 has antinociceptive activity.
• CAS Number: [1838622-25-5]
• MW: 352.4188
• SMILES: FC1C([H])=C([H])C(=C([H])C=1C([H])([H])C([H])([H])N1C([H])([H])C([H])([H])C2(C([H])([H])N(C([H])([H])C([H])([H])[H])C([C@@]([H])(C([H])([H])[H])O2)=O)C([H])([H])C1([H])[H])F
• Formula: C₁₉H₂₆F₂N₂O₂
• Note: For research use only
• Expiration Date: 12 months from date of receipt.