EST73502 hydrochloride

• Catalog Number: orb1685246
• Category: Small Molecules
• Description: EST73502 hydrochloride
• CAS Number: 2535970-65-9
• MW: 388.88
• SMILES: Cl.CCN1CC2(CCN(CCc3cc(F)ccc3F)CC2)O[C@H](C)C1=O
• Formula: C₁₉H₂₇ClF₂N₂O₂
• Biological Activity: EST73502 hydrochloride is a selective, orally active and blood-brain barrier (BBB) penetrant dual μ-opioid receptor (MOR) agonist and σ1 receptor (σ1R) antagonist, with K i s of 64 nM and 118 nM for MOR and σ1R, respectively. EST73502 hydrochloride has antinociceptive activity with reduced opioid-induced relevant adverse events[1].
• Note: For research use only
• Expiration Date: 12 months from date of receipt.