Dersimelagon

• Catalog Number: orb1089631
• Category: Small Molecules
• Description: Dersimelagon, also known as MT-7117 and WHO 10832, is a novel, orally-administered, small molecule, selective melanocortin-1 receptor (MC1R) agonist that increases skin melanin without sun exposure and is being developed to increase light tolerance in EPP/XLP patients. Dersimelagon significantly boosted sunlight tolerance in patients with erythropoietic protoporphyria in a multicenter, phase 2, randomized trial.
• CAS Number: [1835256-48-8]
• MW: 675.7532241
• SMILES: F[C@]1(C(N2C[C@@H](COC)[C@H](C3=CC=C(C(F)(F)F)C=C3N3CCC(C(=O)O)CC3)C2)=O)CN(C[C@@H]1C1C=CC(=CC=1)OC)C1CCCC1
• Formula: C₃₆H₄₅F₄N₃O₅
• Note: For research use only
• Expiration Date: 12 months from date of receipt.