dBET57

• Catalog Number: orb573445
• Category: Small Molecules
• Description: dBET57 is a novel BRD4 heterobifunctional small-molecule ligand (PROTAC), exhibits significant and selective degradation of BRD4 BD1 (DC50/5h=500 nM), but is inactive on BRD4 BD2..
• CAS Number: [1883863-52-2]
• MW: 699.183
• SMILES: CC1=C(SC2=C1C(=N[C@H](C3=NN=C(N32)C)CC(=O)NCCNC4=CC=CC5=C4C(=O)N(C5=O)C6CCC(=O)NC6=O)C7=CC=C(C=C7)Cl)C
• Formula: C₃₄H₃₁ClN₈O₅S
• Note: For research use only
• Expiration Date: 12 months from date of receipt.