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Dbet57

Dbet57

Catalog Number: orb1301789

DispatchUsually dispatched within 3-5 working days
$ 150.00
Catalog Numberorb1301789
CategorySmall Molecules
DescriptionDbet57
CAS Number1883863-52-2
Purity99.52%
MW699.18
SMILESCC=1C2=C(N3C([C@H](CC(NCCNC4=C5C(C(=O)N(C5=O)C6C(=O)NC(=O)CC6)=CC=C4)=O)N=C2C7=CC=C(Cl)C=C7)=NN=C3C)SC1C
FormulaC34H31ClN8O5S
Biological ActivitydBET57 is heterobifunctional degrader of BRD4 based on the PROTAC technology, exhibits significant degradation of BRD4BD1 with a DC50/5h of 500 nM ,and inactive on BRD4BD2
Storage-20°C
NoteFor research use only
Expiration Date12 months from date of receipt.
  • dBET57 [orb573445]

    [1883863-52-2]

    699.183

    C34H31ClN8O5S

    1 g, 100 mg, 250 mg