CYN 154806 TFA

SKU: orb1296646

Description

CYN 154806 TFA is a cyclic octapeptide functioning as a potent and selective somatostatin sst2 receptor antagonist, with pIC50 values of 8.58 (sst2), 5.41 (sst1), 6.07 (sst3), 5.76 (sst4), and 6.48 (sst5). It is a valuable research tool for investigating sst2 receptor function in both in vitro binding assays and in vivo physiological studies.

Research Area

Pharmacology & Drug Discovery

Key Properties

• CAS Number: 2828432-46-6
• MW: 1311.36
• Purity: 99.70% (May vary between batches)
• Formula: C₅₈H₆₉F₃N₁₂O₁₆S₂
• SMILES: C[C@@H](O)[C@H]1C(N[C@H](C(N[C@@H](C(N)=O)CC2=CC=C(O)C=C2)=O)CSSC[C@@H](NC([C@@H](NC(C)=O)CC3=CC=C([N+]([O-])=O)C=C3)=O)C(N[C@@H](CC4=CC=C(O)C=C4)C(N[C@H](CC5=CNC6=CC=CC=C65)C(N[C@@H](CCCCN)C(N1)=O)=O)=O)=O)=O.OC(C(F)(F)F)=O
• Target: Somatostatin
• Solubility: H2O:50 mg/mL (38.13 mM)

Storage & Handling

• Storage: keep away from moisture | Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice/Shipping at ambient temperature.
• Expiration Date: 12 months from date of receipt.
• Disclaimer: For research use only

Alternative Names

CYN 154806 TFA, CYN 154806 TFA(183658 72 2 free base), CYN 154806 TFA(183658722 free base), Somatostatin Receptor

Compound Identifiers

PubChem CID

71312046