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Catalog Number | orb1296646 |
---|---|
Category | Small Molecules |
Description | CYN 154806 TFA(183658-72-2 free base) |
CAS Number | 2828432-46-6 |
Purity | 99.70% |
MW | 1311.36 |
SMILES | C[C@@H](O)[C@H]1C(N[C@H](C(N[C@@H](C(N)=O)CC2=CC=C(O)C=C2)=O)CSSC[C@@H](NC([C@@H](NC(C)=O)CC3=CC=C([N+]([O-])=O)C=C3)=O)C(N[C@@H](CC4=CC=C(O)C=C4)C(N[C@H](CC5=CNC6=CC=CC=C65)C(N[C@@H](CCCCN)C(N1)=O)=O)=O)=O)=O.OC(C(F)(F)F)=O |
Formula | C58H69F3N12O16S2 |
Biological Activity | CYN 154806 TFA is a cyclic octapeptide and an effective selective somatostatin sst2 receptor antagonist. For the recombinant sst2, sst1, sst3, sst4 and sst5 receptors, the pIC50 values are 8.58, 5.41, 6.07, 5.76 and 6.48, respectively. |
Storage | Store at -20°C for 12 months. |
Note | For research use only |
Expiration Date | 12 months from date of receipt. |
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