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Catalog Number | orb1298859 |
---|---|
Category | Small Molecules |
Description | CPYPP |
CAS Number | 310460-39-0 |
Purity | 99.85% |
MW | 324.76 |
SMILES | O=C1N(NC(=O)C1=CC=CC2=C(Cl)C=CC=C2)C3=CC=CC=C3 |
Formula | C18H13ClN2O2 |
Biological Activity | CPYPP is an inhibitor of DOCK2-Rac1 interaction. CPYPP binds to DOCK2 DHR-2 domain and inhibits the guanine nucleotide exchange factor (GEF) activity of DOCK2DHR-2 for Rac1 in a dose-dependent manner(IC50 : 22.8 μM). CPYPP also inhibits DOCK180, DOCK5 and less DOCK9 |
Storage | Store at -20°C for 12 months. |
Note | For research use only |
Expiration Date | 12 months from date of receipt. |
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