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Catalog Number | orb1710011 |
---|---|
Category | Small Molecules |
Description | CNX-500 |
CAS Number | 1202758-21-1 |
Purity | 98% |
MW | 961.18 |
SMILES | C(CCCC(NCCCOCCOCCOCCCNC(CCCC(NCCCOC1=CC(NC=2N=C(NC3=CC(NC(C=C)=O)=CC=C3)C(C)=CN2)=CC=C1)=O)=O)=O)[C@H]4[C@@]5([C@](CS4)(NC(=O)N5)[H])[H] |
Formula | C48H68N10O9S |
Biological Activity | CNX-500 is a probe consisting of a covalent Btk inhibitor chemically linked to biotin. CNX-500 has inhibitory activity against Btk (IC50: 0.5 nM) and the ability to form a covalent bond with Btk. CNX-500 has low inhibitory effects on kinase EGFR and upstream Src-family kinases. |
Storage | Store at -20°C for 12 months. |
Note | For research use only |
Expiration Date | 12 months from date of receipt. |
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