CNX-500

• Catalog Number: orb1710011
• Category: Small Molecules
• Description: CNX-500
• CAS Number: 1202758-21-1
• Purity: 98%
• MW: 961.18
• SMILES: C(CCCC(NCCCOCCOCCOCCCNC(CCCC(NCCCOC1=CC(NC=2N=C(NC3=CC(NC(C=C)=O)=CC=C3)C(C)=CN2)=CC=C1)=O)=O)=O)[C@H]4[C@@]5([C@](CS4)(NC(=O)N5)[H])[H]
• Formula: C₄₈H₆₈N₁₀O₉S
• Biological Activity: CNX-500 is a probe consisting of a covalent Btk inhibitor chemically linked to biotin. CNX-500 has inhibitory activity against Btk (IC50: 0.5 nM) and the ability to form a covalent bond with Btk. CNX-500 has low inhibitory effects on kinase EGFR and upstream Src-family kinases.
• Storage: Store at -20°C for 12 months.
• Note: For research use only
• Expiration Date: 12 months from date of receipt.