CH5447240

• Catalog Number: orb1702427
• Category: Small Molecules
• Description: CH5447240
• CAS Number: 1253919-92-4
• Purity: 98%
• MW: 517.68
• SMILES: O=C1C2(NC(=N1)[C@H]3CC[C@H](C)CC3)CCN(S(CCC4=C(C)C=C(N(C(N)=O)C)C=C4C)(=O)=O)CC2
• Formula: C₂₆H₃₉N₅O₄S
• Biological Activity: CH5447240 is an effective Human Parathyroid Hormone Receptor 1 (hPTHR1) Agonist for the treatment of Hypoparathyroidism. CH5447240 showed a potent in vitro hPTHR1 agonist effect (EC20: 3.0 nM; EC50: 12 nM). It showed 55% oral bioavailability and a significantly elevated serum calcium level in hypocalcemic model rats.
• Storage: Store at -20°C for 12 months.
• Note: For research use only
• Expiration Date: 12 months from date of receipt.