BX795

• Catalog Number: orb1307362
• Category: Small Molecules
• Description: BX795
• CAS Number: 702675-74-9
• Purity: 98.32%
• MW: 591.47
• SMILES: IC1=CN=C(NC2=CC(NC(=O)N3CCCC3)=CC=C2)N=C1NCCCNC(=O)C1=CC=CS1
• Formula: C₂₃H₂₆IN₇O₂S
• Biological Activity: BX795 is an effective and selective PDK1 inhibitor (IC50: 6 nM), and its selectivity is 140- and 1600-fold for PDK1 over PKA and PKC in cell-free assays, respectively. Meanwhile, the selectivity for PDK1 is 100-fold than GSK3β.
• Storage: Store at -20°C for 12 months.
• Note: For research use only
• Expiration Date: 12 months from date of receipt.