Brilaroxazine

• Catalog Number: orb1308521
• Category: Small Molecules
• Description: Brilaroxazine
• CAS Number: 1239729-06-6
• Purity: 98%
• MW: 450.36
• SMILES: O(CCCCN1CCN(CC1)C2=C(Cl)C(Cl)=CC=C2)C=3C=C4C(=CC3)OCC(=O)N4
• Formula: C₂₂H₂₅Cl₂N₃O₃
• Biological Activity: Brilaroxazine (RP5063) is a potent multimodal dopamine/5-HT modulator. Brilaroxazine is a partial agonist of dopamine D2, D3, and D4 receptors, 5-HT1A (Ki =1.5 nM) and 5-HT2A (Ki = 2.5 nM), and has antagonist activity 5-HT2B, and 5-HT7 receptors with Kis of 0.19 nM and 2.7 nM, respectively. Brilaroxazine can be used for research about cognitive impairments in neuropsychiatric and neurological diseases.
• Storage: Store at -20°C for 12 months.
• Note: For research use only
• Expiration Date: 12 months from date of receipt.