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    Borussertib

    Borussertib

    Catalog Number: orb1298943

    DispatchUsually dispatched within 3-5 working days
    $ 1,480.00
    Catalog Numberorb1298943
    CategorySmall Molecules
    DescriptionBorussertib
    CAS Number1800070-77-2
    Purity98.18%
    MW596.68
    SMILESO=C1N(C=2C(N1)=CC=C(NC(C=C)=O)C2)C3CCN(CC4=CC=C(C=C4)C5=C(C=C6C(=N5)C=CNC6=O)C7=CC=CC=C7)CC3
    FormulaC36H32N6O3
    Biological ActivityBorussertib is a covalent-allosteric and first-in-class inhibitor of protein kinase Akt(IC50 of 0.8 nM and a Ki of 2.2 nM for Aktwt)
    StorageStore at -20°C for 12 months.
    NoteFor research use only
    Expiration Date12 months from date of receipt.
    • Borussertib [orb654596]

      [1800070-77-2]

      596.691

      C36H32N6O3

      1 g, 100 mg, 250 mg
    • Borussertib [orb1897044]

      1800070-77-2

      50 mg
    • Borussertib [orb1897045]

      1800070-77-2

      5 mg
    • Borussertib [orb1897046]

      1800070-77-2

      100 mg
    • Borussertib [orb1897047]

      1800070-77-2

      10 mg
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