BKI1369

• Catalog Number: orb654579
• Category: Small Molecules
• Description: BKI-1369 is a bumped kinase inhibitor (BKI). BKI-1369 increases human Ether-a-go-go-related gene (hERG)-inhibitory activity with an IC50 of 1.52 μM. BKI-1369 reduces the parasite burden and diseases severity in the gnotobiotic pig model. BKI-1369 has been well characterized for potency, stability, metabolism, toxicity, pharmacokinetics and is potent against C. parvum in infected mice and calves.
• CAS Number: [1951431-22-3]
• MW: 417.51
• SMILES: NC1N=CN=C2N(N=C(C3C=C4C(N=C(C=C4)OCC)=CC=3)C=12)CC1CCN(C)CC1
• Formula: C₂₃H₂₇N₇O
• Note: For research use only
• Expiration Date: 12 months from date of receipt.