β2AR/M-receptor agonist-2

• Catalog Number: orb1745044
• Category: Small Molecules
• Description: β2AR/M-receptor agonist-2
• CAS Number: 1017857-38-3
• MW: 717.31
• SMILES: N(C(OC1CCN(CCCCCCCCCNC[C@H](O)C2=CC(NS(C)(=O)=O)=C(O)C=C2)CC1)=O)C3=C(C=CC=C3)C4=CC(Cl)=C(O)C=C4
• Formula: C₃₆H₄₉ClN₄O₇S
• Biological Activity: β2AR/M-receptor agonist-2 is a dual-function compound acting as a muscarinic antagonist and β2 adrenoceptor agonist (MABA). It demonstrates significant activity towards the β2 adrenoceptor with an EC50 of 3.7 nM and exhibits affinity for the human cloned M3 receptor with a Ki of 0.73 nM. This potent bronchodilator holds potential for research in chronic obstructive pulmonary disease (COPD) treatment.
• Storage: Store at -20°C for 12 months.
• Note: For research use only
• Expiration Date: 12 months from date of receipt.