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Catalog Number | orb1982697 |
---|---|
Category | Small Molecules |
Description | β2AR/M-receptor agonist-1 |
CAS Number | 2230520-62-2 |
MW | 806.82 |
SMILES | [Br-].O[C@H](CNCCCOc1ccc(OCCC[N+]23CCC(CC2)[C@@H](C3)OC[C@@](O)(C2CCCC2)c2ccccc2)cc1)c1ccc(O)c2[nH]c(=O)ccc12 |
Formula | C43H56BrN3O7 |
Biological Activity | β2AR/M-receptor agonist-1 (example 131), a muscarinic antagonist and β2 adrenoceptor agonist (MABA), exhibits dual potency towards β2 adrenoceptor and muscarinic receptor. It demonstrates a significant affinity for the β2 adrenoceptor, indicated by an EC50 value of 9.2 nM, and for the muscarinic receptor with a Ki value of 30.2 nM. Furthermore, its MABA activity is highlighted by an EC50 value of 4.0 nM [1]. |
Storage | Store at -20°C for 12 months. |
Note | For research use only |
Expiration Date | 12 months from date of receipt. |
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