β2AR/M-receptor agonist-1

• Catalog Number: orb1982697
• Category: Small Molecules
• Description: β2AR/M-receptor agonist-1
• CAS Number: 2230520-62-2
• MW: 806.82
• SMILES: [Br-].O[C@H](CNCCCOc1ccc(OCCC[N+]23CCC(CC2)[C@@H](C3)OC[C@@](O)(C2CCCC2)c2ccccc2)cc1)c1ccc(O)c2[nH]c(=O)ccc12
• Formula: C₄₃H₅₆BrN₃O₇
• Biological Activity: β2AR/M-receptor agonist-1 (example 131), a muscarinic antagonist and β2 adrenoceptor agonist (MABA), exhibits dual potency towards β2 adrenoceptor and muscarinic receptor. It demonstrates a significant affinity for the β2 adrenoceptor, indicated by an EC50 value of 9.2 nM, and for the muscarinic receptor with a Ki value of 30.2 nM. Furthermore, its MABA activity is highlighted by an EC50 value of 4.0 nM [1].
• Storage: Store at -20°C for 12 months.
• Note: For research use only
• Expiration Date: 12 months from date of receipt.